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Results 1-15 of 25 (Search time: 0.005 seconds).
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Issue DateTitleInvolved Person(s)
10-Jun-2019Approaching target selectivity by de novo drug designFischer, Thomas; Gazzola, Silvia; Riedl, Rainer
18-Feb-2019Titelbild: Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐Grundgerüsts (Angew. Chem. 12/2019)Gall, Flavio M.; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
18-Feb-2019Cover picture : drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor template (Angew. Chem. Int. Ed. 12/2019)Gall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
5-Feb-2019Design and structural evolution of matrix metalloproteinase inhibitorsFischer, Thomas; Senn, Nicole; Riedl, Rainer
7-Jan-2019Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐GrundgerüstsGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
7-Jan-2019Drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor templateGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
30-May-2018Eine strukturelle Evaluierung medizinalchemischer Strategien gegen WirkstoffresistenzenAgnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer
30-May-2018A Structural view on medicinal chemistry strategies against drug resistanceAgnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer
2017Emodin : a compound with putative antidiabetic potential, deteriorates glucose tolerance in rodentsAbu Eid, Sameer; Adams, Michael; Scherer, Thomas; Torres-Gómez, Héctor Manuel; Hackl, Martina Theresa; Kaplanian, Mairam; Riedl, Rainer; Luger, Anton; Fürnsinn, Clemens
2017Pseudouridimycin : the first nucleoside analogue that selectively inhibits bacterial RNA polymeraseChellat, Mathieu F.; Riedl, Rainer
2017Targeted polypharmacology : discovery of a highly potent non-hydroxamate dual matrix metalloproteinase (MMP)-10/-13 inhibitorSenn, Nicole; Ott, Michael; Lanz, Jan; Riedl, Rainer
2017Pseudouridimycin : das erste Nukleosid-Analogon, das bakterielle RNA-Polymerase selektiv inhibiertChellat, Mathieu F.; Riedl, Rainer
Sep-2016Emodin, a compound with acclaimed antidiabetic potential, deteriorates glucose tolerance in obese miceAbu Eid, S.; Adams, M.; Scherer, T.; Torres-Gómez, H.; Hackl, M.T.; Riedl, R.; Luger, A.; Fürnsinn, C.
24-Oct-2015Emodin, eine mutmaßlich anti-diabetisch wirksame Verbindung, beeinträchtigt die Glukosetoleranz adipöser MäuseAbu Eud, Sameer; Adams, Michael; Scherer, Thomas; Torres-Gomez, Hector; Riedl, Rainer; Luger, Anton; Fürnsinn, Clemens
25-Feb-2015Cover Picture: Merging allosteric and active site binding motifs : de novo generation of target selectivity and potency via natural‐product‐derived fragments (ChemMedChem 3/2015)Lanz, Jan; Riedl, Rainer
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