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Issue DateTitleInvolved Person(s)
30-Dec-2019CyBy2 : a strongly typed, purely functional framework for chemical data managementHöck, Stefan; Riedl, Rainer
10-Jun-2019Approaching target selectivity by de novo drug designFischer, Thomas; Gazzola, Silvia; Riedl, Rainer
1-May-2019Durch die Natur inspiriertes WirkstoffdesignGall, Flavio; Riedl, Rainer; Sievers, Martin; Wermelinger, Tobias; Frasson, David
18-Feb-2019Titelbild: Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐Grundgerüsts (Angew. Chem. 12/2019)Gall, Flavio M.; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
18-Feb-2019Cover picture : drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor template (Angew. Chem. Int. Ed. 12/2019)Gall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
5-Feb-2019Design and structural evolution of matrix metalloproteinase inhibitorsFischer, Thomas; Senn, Nicole; Riedl, Rainer
7-Jan-2019Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐GrundgerüstsGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
7-Jan-2019Drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor templateGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
2019High consistency of structure-based design and x-ray crystallography : design, synthesis, kinetic evaluation and crystallographic binding mode determination of biphenyl-N-acyl-β-D-glucopyranosylamines as glycogen phosphorylase inhibitorsFischer, Thomas; Koulas, Symeon M.; Tsagkarakou, Anastasia S.; Kyriakis, Efthimios; Stravodimos, George A.; Skamnaki, Vassiliki T.; Liggri, Panagiota G.V.; Zographos, Spyros E.; Riedl, Rainer; Leonidas, Demetres D.
2019Inhibitory antibodies designed for matrix metalloproteinase modulationFischer, Thomas; Riedl, Rainer