Search


Results 1-15 of 55 (Search time: 0.008 seconds).
Item hits:
Issue DateTitleInvolved Person(s)
30-Dec-2019CyBy2 : a strongly typed, purely functional framework for chemical data managementHöck, Stefan; Riedl, Rainer
10-Jun-2019Approaching target selectivity by de novo drug designFischer, Thomas; Gazzola, Silvia; Riedl, Rainer
1-May-2019Durch die Natur inspiriertes WirkstoffdesignGall, Flavio; Riedl, Rainer; Sievers, Martin; Wermelinger, Tobias; Frasson, David
18-Feb-2019Titelbild: Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐Grundgerüsts (Angew. Chem. 12/2019)Gall, Flavio M.; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
18-Feb-2019Cover picture : drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor template (Angew. Chem. Int. Ed. 12/2019)Gall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
5-Feb-2019Design and structural evolution of matrix metalloproteinase inhibitorsFischer, Thomas; Senn, Nicole; Riedl, Rainer
7-Jan-2019Von der Natur inspiriertes Wirkstoffdesign : kristallographische Detektion eines selbstgenerierten Inhibitor‐GrundgerüstsGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
7-Jan-2019Drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor templateGall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E.; Sievers, Martin; Riedl, Rainer
2019High consistency of structure-based design and x-ray crystallography : design, synthesis, kinetic evaluation and crystallographic binding mode determination of biphenyl-N-acyl-β-D-glucopyranosylamines as glycogen phosphorylase inhibitorsFischer, Thomas; Koulas, Symeon M.; Tsagkarakou, Anastasia S.; Kyriakis, Efthimios; Stravodimos, George A.; Skamnaki, Vassiliki T.; Liggri, Panagiota G.V.; Zographos, Spyros E.; Riedl, Rainer; Leonidas, Demetres D.
2019Inhibitory antibodies designed for matrix metalloproteinase modulationFischer, Thomas; Riedl, Rainer
5-Oct-2018Primary resistance mechanism of the canine distemper virus fusion protein against a small-molecule membrane fusion inhibitorKalbermatter, David; Shrestha, Neeta; Ader-Ebert, Nadine; Herren, Michael; Moll, Pascal; Plemper, Richard K.; Altmann, Karl-Heinz; Langedijk, Johannes P.; Gall, Flavio; Lindenmann, Urs; Riedl, Rainer; Fotiadis, Dimitrios; Plattet, Philippe
11-Jul-2018Antiprotozoal compoundsAgnello, Stefano; Adams, Michael; Kaiser, Marcel; Mäser, Pascal; Urban, Alexander; Raguz, Luka; Riedl, Rainer
30-May-2018Eine strukturelle Evaluierung medizinalchemischer Strategien gegen WirkstoffresistenzenAgnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer
30-May-2018A Structural view on medicinal chemistry strategies against drug resistanceAgnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer
2017Emodin : a compound with putative antidiabetic potential, deteriorates glucose tolerance in rodentsAbu Eid, Sameer; Adams, Michael; Scherer, Thomas; Torres-Gómez, Héctor Manuel; Hackl, Martina Theresa; Kaplanian, Mairam; Riedl, Rainer; Luger, Anton; Fürnsinn, Clemens
Results 1-15 of 55 (Search time: 0.008 seconds).