Issue Date | Title | Involved Person(s) |
7-Jan-2019 | Drug design inspired by nature : crystallographic detection of an auto‐tailored protease inhibitor template | Gall, Flavio; Hohl, Deborah; Frasson, David; Wermelinger, Tobias; Mittl, Peer R. E., et al |
2019 | High consistency of structure-based design and x-ray crystallography : design, synthesis, kinetic evaluation and crystallographic binding mode determination of biphenyl-N-acyl-β-D-glucopyranosylamines as glycogen phosphorylase inhibitors | Fischer, Thomas; Koulas, Symeon M.; Tsagkarakou, Anastasia S.; Kyriakis, Efthimios; Stravodimos, George A., et al |
2019 | Inhibitory antibodies designed for matrix metalloproteinase modulation | Fischer, Thomas; Riedl, Rainer |
5-Oct-2018 | Primary resistance mechanism of the canine distemper virus fusion protein against a small-molecule membrane fusion inhibitor | Kalbermatter, David; Shrestha, Neeta; Ader-Ebert, Nadine; Herren, Michael; Moll, Pascal, et al |
11-Jul-2018 | Antiprotozoal compounds | Agnello, Stefano; Adams, Michael; Kaiser, Marcel; Mäser, Pascal; Urban, Alexander, et al |
30-May-2018 | Eine strukturelle Evaluierung medizinalchemischer Strategien gegen Wirkstoffresistenzen | Agnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer |
30-May-2018 | A Structural view on medicinal chemistry strategies against drug resistance | Agnello, Stefano; Brand, Michael; Chellat, Mathieu; Gazzola, Silvia; Riedl, Rainer |
2017 | Emodin : a compound with putative antidiabetic potential, deteriorates glucose tolerance in rodents | Abu Eid, Sameer; Adams, Michael; Scherer, Thomas; Torres-Gómez, Héctor Manuel; Hackl, Martina Theresa, et al |
2017 | Development of a non-hydroxamate dual matrix metalloproteinase (MMP)-7/-13 inhibitor | Fischer, Thomas; Riedl, Rainer |
2017 | Cover profile : targeted fluoro positioning for the discovery of a potent and highly selective matrix metalloproteinase inhibitor | Fischer, Thomas; Riedl, Rainer |
2017 | Pseudouridimycin : the first nucleoside analogue that selectively inhibits bacterial RNA polymerase | Chellat, Mathieu F.; Riedl, Rainer |
2017 | Cover picture : targeted fluoro positioning for the discovery of a potent and highly selective matrix metalloproteinase inhibitor (ChemistryOpen 2/2017) | Fischer, Thomas; Riedl, Rainer |
2017 | Targeted polypharmacology : discovery of a highly potent non-hydroxamate dual matrix metalloproteinase (MMP)-10/-13 inhibitor | Senn, Nicole; Ott, Michael; Lanz, Jan; Riedl, Rainer |
2017 | Targeted fluoro positioning for the discovery of a potent and highly selective matrix metalloproteinase inhibitor | Fischer, Thomas; Riedl, Rainer |
2017 | Pseudouridimycin : das erste Nukleosid-Analogon, das bakterielle RNA-Polymerase selektiv inhibiert | Chellat, Mathieu F.; Riedl, Rainer |